THIOGUANINE ANHYDROUS: 1,168 Adverse Event Reports & Safety Profile
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1,168
Total FAERS Reports
175 (15.0%)
Deaths Reported
599
Hospitalizations
1,168
As Primary/Secondary Suspect
77
Life-Threatening
12
Disabilities
First Report: 1995 · Latest Report: 20250610
What Are the Most Common THIOGUANINE ANHYDROUS Side Effects?
#1 Most Reported
Febrile neutropenia
191 reports (16.4%)
#2 Most Reported
Off label use
98 reports (8.4%)
#3 Most Reported
Venoocclusive liver disease
85 reports (7.3%)
All THIOGUANINE ANHYDROUS Side Effects by Frequency
| Side Effect | Reports | % of Total | Deaths | Hosp. |
|---|---|---|---|---|
| Febrile neutropenia | 191 | 16.4% | 26 | 147 |
| Off label use | 98 | 8.4% | 11 | 35 |
| Venoocclusive liver disease | 85 | 7.3% | 6 | 26 |
| Pancytopenia | 74 | 6.3% | 17 | 63 |
| Pyrexia | 72 | 6.2% | 9 | 66 |
| Drug ineffective | 69 | 5.9% | 11 | 40 |
| Thrombocytopenia | 63 | 5.4% | 10 | 45 |
| Anaemia | 62 | 5.3% | 9 | 36 |
| Neutropenia | 54 | 4.6% | 4 | 43 |
| Abdominal pain | 53 | 4.5% | 2 | 21 |
| Pancreatitis | 53 | 4.5% | 0 | 26 |
| Febrile bone marrow aplasia | 48 | 4.1% | 0 | 48 |
| Vomiting | 43 | 3.7% | 3 | 40 |
| Therapeutic product effect decreased | 42 | 3.6% | 0 | 18 |
| Diarrhoea | 41 | 3.5% | 2 | 20 |
| Leukopenia | 41 | 3.5% | 8 | 21 |
| Venoocclusive disease | 40 | 3.4% | 22 | 17 |
| Drug interaction | 39 | 3.3% | 0 | 7 |
| Fatigue | 38 | 3.3% | 0 | 18 |
| Multiple organ dysfunction syndrome | 37 | 3.2% | 32 | 9 |
Who Reports THIOGUANINE ANHYDROUS Side Effects? Age & Gender Data
Gender: 44.8% female, 55.2% male. Average age: 16.7 years. Most reports from: US. View detailed demographics →
Is THIOGUANINE ANHYDROUS Getting Safer? Reports by Year
| Year | Reports | Deaths | Hosp. |
|---|---|---|---|
| 2000 | 7 | 0 | 0 |
| 2010 | 3 | 0 | 0 |
| 2012 | 6 | 0 | 0 |
| 2013 | 11 | 1 | 8 |
| 2014 | 41 | 2 | 27 |
| 2015 | 14 | 1 | 6 |
| 2016 | 35 | 5 | 22 |
| 2017 | 189 | 5 | 138 |
| 2018 | 112 | 4 | 87 |
| 2019 | 41 | 2 | 36 |
| 2020 | 21 | 1 | 17 |
| 2021 | 45 | 4 | 35 |
| 2022 | 71 | 5 | 61 |
| 2023 | 15 | 1 | 9 |
| 2024 | 2 | 0 | 1 |
| 2025 | 19 | 1 | 15 |
What Is THIOGUANINE ANHYDROUS Used For?
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Official FDA Label for THIOGUANINE ANHYDROUS
Official prescribing information from the FDA-approved drug label.