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Important: This site presents data from the FDA Adverse Event Reporting System (FAERS). A report does not mean the drug caused the event. Full disclaimer.

Transgender hormonal therapy: Which Medications Are Safest? (42 Drugs Compared)

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42 medications are used for Transgender hormonal therapy, with 936 combined adverse event reports. The most reported drugs for Transgender hormonal therapy are TESTOSTERONE and ESTRADIOL.

936
Total Reports
42
Drugs Used

All Medications for Transgender hormonal therapy Ranked by Safety Reports

Drug Brand Reports Deaths (all) Hosp. (all) Death Rate
TESTOSTERONE Testosterone 384 1,091 5,432 4.0%
ESTRADIOL Estradiol 282 267 1,953 0.9%
TESTOSTERONE CYPIONATE Testosterone Cypionate 114 230 1,826 4.4%
CYPROTERONE - 85 42 296 5.4%
LEUPROLIDE Fensolvi 55 11,858 10,499 16.7%
TESTOSTERONE UNDECANOATE Tlando 47 32 193 2.0%
SPIRONOLACTONE spironolactone 36 1,809 11,611 8.6%
PROGESTERONE Progesterone 18 222 1,143 4.0%
TESTOSTERONE ENANTHATE XYOSTED 18 167 457 9.9%
ESTROGENS, CONJUGATED Premarin 16 171 892 1.9%
MEDROXYPROGESTERONE Provera 15 135 831 1.6%
TRIPTORELIN TRIPTODUR 15 528 1,315 9.8%
FINASTERIDE Finasteride 14 524 2,086 3.4%
BICALUTAMIDE Bicalutamide 10 462 1,486 11.4%
ESTROGENS - 8 42 92 12.1%
METHYLTESTOSTERONE METHITEST 5 13 49 17.3%

View all 42 drugs →

Most Reported Drugs for Transgender hormonal therapy

#1 most reported
#2 most reported
#3 most reported