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Important: This site presents data from the FDA Adverse Event Reporting System (FAERS). A report does not mean the drug caused the event. Full disclaimer.

All Drugs Associated with Off label use

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3,309 drugs have been associated with Off label use in FAERS reports.

Drug Reports Deaths Hosp. Life-Threat.
RITUXIMAB 39,751 6,335 11,201 4,207
INFLIXIMAB 34,801 2,600 9,509 2,818
DENOSUMAB 34,612 299 730 55
METHOTREXATE 24,020 3,417 7,881 3,680
VEDOLIZUMAB 21,017 637 5,998 256
ETANERCEPT 20,178 1,852 4,129 2,209
TOCILIZUMAB 18,256 3,347 5,844 2,763
PREDNISONE 17,867 3,499 6,978 3,057
LENALIDOMIDE 17,017 1,252 3,116 250
ADALIMUMAB 16,417 2,187 5,051 2,662
HYDROXYCHLOROQUINE 15,318 2,584 5,688 2,773
INFLIXIMAB-DYYB 14,256 274 3,718 71
MYCOPHENOLATE MOFETIL 13,474 2,365 4,340 1,474
DEXAMETHASONE 13,439 2,704 4,927 1,297
CYCLOPHOSPHAMIDE 12,578 2,788 3,928 1,159
RUXOLITINIB 12,492 1,527 1,769 111
BEVACIZUMAB 12,094 3,560 1,814 227
TOFACITINIB 11,736 1,767 3,218 2,094
ABATACEPT 10,990 1,752 3,770 2,430
USTEKINUMAB 10,990 1,395 2,924 1,779
DUPILUMAB 10,543 54 291 12
RISPERIDONE 10,376 245 1,621 182
DICLOFENAC 10,370 1,995 2,649 2,336
METHYLPREDNISOLONE 10,364 2,842 4,839 2,315
CERTOLIZUMAB PEGOL 10,281 1,629 3,112 2,024
ONABOTULINUMTOXINA 9,698 181 331 70
ACETAMINOPHEN 9,410 2,262 3,754 2,429
LEFLUNOMIDE 9,265 2,125 3,934 2,748
OMALIZUMAB 9,199 100 627 123
PREDNISOLONE 8,817 1,617 3,586 1,001
GOLIMUMAB 8,764 1,664 3,186 2,017
TACROLIMUS 8,718 1,378 3,230 735
DOXORUBICIN 7,858 1,712 2,385 732
CETIRIZINE 7,790 1,836 2,578 2,182
SULFASALAZINE 7,626 1,692 3,213 2,331
TIRZEPATIDE 7,007 21 425 30
CYCLOSPORINE 6,860 1,043 1,817 461
INSULIN GLARGINE 6,842 21 317 44
GABAPENTIN 6,729 530 1,510 357
VINCRISTINE 6,562 1,506 1,919 610
ETOPOSIDE 6,495 1,541 2,054 776
VENETOCLAX 6,252 2,257 1,642 110
CARBOPLATIN 6,100 957 2,160 561
HUMAN IMMUNOGLOBULIN G 5,872 787 1,808 455
LEVETIRACETAM 5,789 456 2,040 383
PREGABALIN 5,713 840 1,935 795
APIXABAN 5,590 491 1,869 337
SECUKINUMAB 5,566 1,926 2,601 2,293
ARIPIPRAZOLE 5,473 202 2,042 236
IBRUTINIB 5,446 866 1,760 120
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