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Important: This site presents data from the FDA Adverse Event Reporting System (FAERS). A report does not mean the drug caused the event. Full disclaimer.

All Drugs Associated with Off label use (Page 4)

3,309 drugs have been associated with Off label use in FAERS reports.

Drug Reports Deaths Hosp. Life-Threat.
RITUXIMAB-PVVR 2,079 209 502 48
VANCOMYCIN 2,070 506 1,095 308
LEUPROLIDE 2,060 73 221 19
CHLORHEXIDINE 2,055 1,291 1,567 1,434
RAMIPRIL 2,053 1,151 1,531 1,176
SARILUMAB 2,035 824 933 1,016
TRIAMCINOLONE ACETONIDE 2,034 812 1,314 927
IRINOTECAN 2,018 345 630 119
LOPINAVIR\RITONAVIR 2,010 370 798 111
MELPHALAN 2,002 437 495 243
SIROLIMUS 1,960 251 523 124
FENTANYL 1,958 170 725 193
BUPRENORPHINE\NALOXONE 1,946 18 179 15
COPPER 1,941 0 12 0
FILGRASTIM 1,930 387 578 110
CANDESARTAN 1,911 967 1,124 981
GOLD THIOMALATE 1,909 904 1,394 983
REGORAFENIB 1,906 244 702 34
ONDANSETRON 1,905 449 658 267
PERTUZUMAB 1,886 373 655 63
VALGANCICLOVIR 1,882 376 578 81
LURASIDONE 1,878 32 309 33
BUPRENORPHINE 1,868 835 937 744
SERTRALINE 1,865 122 661 99
AMLODIPINE 1,835 234 845 246
BOTULINUM TOXIN TYPE A 1,785 786 847 714
DOCETAXEL 1,782 410 745 110
CIPROFLOXACIN 1,781 225 852 121
LINEZOLID 1,781 326 782 185
ALTEPLASE 1,752 137 135 36
ISOTRETINOIN 1,731 19 95 16
FLUMETHASONE PIVALATE 1,718 1,172 1,401 1,503
ENOXAPARIN 1,707 237 679 115
MIRABEGRON 1,704 722 705 661
PEMETREXED 1,663 308 652 143
CODEINE 1,662 258 546 168
ATORVASTATIN 1,654 98 868 61
CANNABIDIOL 1,636 185 770 17
DOXYCYCLINE 1,630 375 756 446
ALPRAZOLAM 1,614 179 665 93
HUMAN C1-ESTERASE INHIBITOR 1,614 808 964 784
AMIODARONE 1,608 513 872 448
GOLD 1,601 578 989 648
ROSUVASTATIN 1,594 29 554 110
AMITRIPTYLINE 1,588 72 435 145
SORAFENIB 1,587 301 563 38
DARBEPOETIN ALFA 1,586 364 446 124
PIPERACILLIN\TAZOBACTAM 1,586 398 902 291
LEVOTHYROXINE 1,585 130 578 214
OBINUTUZUMAB 1,584 139 239 43
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