Cytochrome P450 3A Inhibitors [MoA]: Side Effects & Safety Data for 31 Drugs
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Cytochrome P450 3A Inhibitors [MoA] includes 31 drugs with a combined 377,767 adverse event reports in the FDA FAERS database. Compare their safety profiles, side effects, and outcomes below.
31
Drugs in Class
377,767
Combined Reports
All Cytochrome P450 3A Inhibitors [MoA] Drugs Ranked by Reports
| Drug | Brand Name | Reports | Deaths | Hosp. | Death Rate |
|---|---|---|---|---|---|
| PALBOCICLIB | Ibrance | 91,024 | 11,066 | 13,442 | 12.2% |
| AMLODIPINE | Olmesartan Medoxomil, Amlodipine and Hydrochlorothiazide | 64,924 | 10,161 | 26,787 | 15.7% |
| RIBOCICLIB | KISQALI | 27,997 | 4,501 | 6,700 | 16.1% |
| OSIMERTINIB | TAGRISSO | 27,750 | 12,456 | 5,277 | 44.9% |
| AMIODARONE | Amiodarone Hydrochloride | 25,143 | 3,845 | 13,711 | 15.3% |
| MIRABEGRON | MIRABEGRON | 20,618 | 1,338 | 2,589 | 6.5% |
| CLARITHROMYCIN | Clarithromycin | 18,945 | 987 | 6,385 | 5.2% |
| RITONAVIR | Norvir | 11,980 | 1,190 | 2,925 | 9.9% |
| CRIZOTINIB | Xalkori | 9,948 | 3,173 | 2,520 | 31.9% |
| RANOLAZINE | Ranolazine | 9,522 | 1,048 | 3,367 | 11.0% |
| SUVOREXANT | BELSOMRA | 9,413 | 219 | 572 | 2.3% |
| VERAPAMIL | Verapamil Hydrochloride | 9,320 | 2,630 | 3,576 | 28.2% |
| IDELALISIB | Zydelig | 6,862 | 1,548 | 2,962 | 22.6% |
| IVACAFTOR | Kalydeco | 6,735 | 291 | 3,756 | 4.3% |
| TUCATINIB | TUKYSA | 6,042 | 640 | 1,717 | 10.6% |
| CENOBAMATE | Xcopri | 5,643 | 125 | 1,012 | 2.2% |
| ATAZANAVIR | Atazanavir Sulfate | 5,434 | 425 | 1,112 | 7.8% |
| DARUNAVIR ETHANOLATE | PREZISTA | 4,389 | 397 | 1,069 | 9.0% |
| DARUNAVIR | Darunavir | 3,558 | 433 | 841 | 12.2% |
| CERITINIB | ZYKADIA | 2,796 | 786 | 804 | 28.1% |
| DRONEDARONE | Multaq | 2,735 | 115 | 611 | 4.2% |
| RITLECITINIB | Litfulo | 1,441 | 1 | 47 | 0.1% |
| LETERMOVIR | PREVYMIS | 1,416 | 252 | 398 | 17.8% |
| NELFINAVIR | VIRACEPT | 1,164 | 87 | 162 | 7.5% |
| SELPERCATINIB | RETEVMO | 1,084 | 160 | 342 | 14.8% |
| LENACAPAVIR | Sunlenca | 502 | 32 | 42 | 6.4% |
| NIROGACESTAT | OGSIVEO | 497 | 7 | 54 | 1.4% |
| PIRTOBRUTINIB | JAYPIRCA | 437 | 130 | 144 | 29.7% |
| COBICISTAT | Tybost | 347 | 41 | 109 | 11.8% |
| LONAFARNIB | Zokinvy | 59 | 6 | 14 | 10.2% |
| TRICLABENDAZOLE | EGATEN | 42 | 0 | 4 | N/A |
Common Side Effects in Cytochrome P450 3A Inhibitors [MoA] Drugs
| Side Effect | Reports | Deaths |
|---|---|---|
| Fatigue | 29,303 | 2,142 |
| Death | 29,071 | 29,002 |
| Nausea | 22,548 | 2,191 |
| Drug ineffective | 20,967 | 1,802 |
| Diarrhoea | 18,437 | 1,737 |
| Dyspnoea | 15,619 | 2,325 |
| Off label use | 14,972 | 2,567 |
| White blood cell count decreased | 13,750 | 592 |
| Dizziness | 13,175 | 1,163 |
| Vomiting | 13,058 | 1,982 |