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Important: This site presents data from the FDA Adverse Event Reporting System (FAERS). A report does not mean the drug caused the event. Full disclaimer.

Protein Kinase Inhibitors [MoA]: Side Effects & Safety Data for 18 Drugs

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Protein Kinase Inhibitors [MoA] includes 18 drugs with a combined 341,716 adverse event reports in the FDA FAERS database. Compare their safety profiles, side effects, and outcomes below.

18
Drugs in Class
341,716
Combined Reports

All Protein Kinase Inhibitors [MoA] Drugs Ranked by Reports

Drug Brand Name Reports Deaths Hosp. Death Rate
IBRUTINIB Imbruvica 75,087 12,580 24,920 16.8%
EVEROLIMUS EVEROLIMUS 39,640 8,374 11,211 21.1%
CABOZANTINIB S-MALATE CABOMETYX 39,270 4,203 6,193 10.7%
DASATINIB dasatinib 30,019 2,681 6,437 8.9%
ERLOTINIB Erlotinib 22,472 6,791 3,693 30.2%
SUNITINIB MALATE Sunitinib malate 21,578 6,028 5,720 27.9%
PAZOPANIB Pazopanib 21,208 5,612 4,347 26.5%
DABRAFENIB Tafinlar 19,305 4,165 5,325 21.6%
TRAMETINIB DIMETHYL SULFOXIDE Mekinist 16,286 3,925 3,438 24.1%
SIROLIMUS sirolimus 11,371 1,737 3,535 15.3%
SORAFENIB sorafenib 10,908 2,489 3,547 22.8%
PONATINIB Iclusig 10,011 2,924 4,254 29.2%
VEMURAFENIB ZELBORAF 8,562 1,040 2,368 12.1%
AFATINIB Gilotrif 6,078 1,346 2,055 22.1%
GEFITINIB Gefitinib 4,697 1,047 853 22.3%
LAPATINIB DITOSYLATE Lapatinib 3,948 921 752 23.3%
VANDETANIB CAPRELSA 1,159 93 363 8.0%
NINTEDANIB ESYLATE Ofev 117 23 39 19.7%

Common Side Effects in Protein Kinase Inhibitors [MoA] Drugs

Side EffectReportsDeaths
Death 41,513 41,428
Diarrhoea 34,613 3,170
Fatigue 28,712 2,423
Off label use 21,593 3,820
Nausea 20,944 1,984
Rash 18,564 1,601
Malignant neoplasm progression 16,760 5,457
Pyrexia 14,428 1,814
Decreased appetite 14,321 1,961
Vomiting 12,162 1,630
View detailed side effects for this class → Compare drugs in this class →