Histamine H1 Receptor Antagonists [MoA]: Side Effects & Safety Data for 13 Drugs
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Histamine H1 Receptor Antagonists [MoA] includes 13 drugs with a combined 133,955 adverse event reports in the FDA FAERS database. Compare their safety profiles, side effects, and outcomes below.
13
Drugs in Class
133,955
Combined Reports
All Histamine H1 Receptor Antagonists [MoA] Drugs Ranked by Reports
| Drug | Brand Name | Reports | Deaths | Hosp. | Death Rate |
|---|---|---|---|---|---|
| CETIRIZINE | Cetirizine | 47,655 | 4,787 | 8,423 | 10.0% |
| DIPHENHYDRAMINE | Allergy Relief | 25,827 | 10,508 | 6,849 | 40.7% |
| FEXOFENADINE | Fexofenadine HCl | 21,453 | 80 | 535 | 0.4% |
| LEVOCETIRIZINE | allergy relief | 10,782 | 554 | 884 | 5.1% |
| OLOPATADINE | PATADAY ONCE DAILY RELIEF | 8,787 | 89 | 171 | 1.0% |
| AZELASTINE | Azelastine Hydrochloride | 5,896 | 12 | 89 | 0.2% |
| KETOTIFEN | Eye Itch Relief | 5,209 | 9 | 99 | 0.2% |
| DESLORATADINE | Desloratadine | 3,141 | 160 | 1,389 | 5.1% |
| DIMENHYDRINATE | Driminate | 1,934 | 160 | 836 | 8.3% |
| CHLORPHENIRAMINE | ACTIDOM DA | 1,919 | 607 | 663 | 31.6% |
| EPINASTINE | EPINASTINE HYDROCHLORIDE | 843 | 6 | 25 | 0.7% |
| ALCAFTADINE | Alcaftadine | 465 | 0 | 4 | N/A |
| CARBINOXAMINE | Carbinoxamine Maleate Extended-Release Oral Suspension | 44 | 3 | 2 | 6.8% |
Common Side Effects in Histamine H1 Receptor Antagonists [MoA] Drugs
| Side Effect | Reports | Deaths |
|---|---|---|
| Drug ineffective | 31,139 | 1,809 |
| Treatment failure | 14,610 | 1,443 |
| Fatigue | 14,309 | 2,706 |
| Pain | 12,244 | 2,224 |
| Off label use | 11,883 | 2,384 |
| Rheumatoid arthritis | 9,708 | 2,437 |
| Abdominal discomfort | 9,669 | 2,183 |
| Alopecia | 9,276 | 2,117 |
| Rash | 9,084 | 2,389 |
| Hypersensitivity | 8,820 | 2,243 |