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Important: This site presents data from the FDA Adverse Event Reporting System (FAERS). A report does not mean the drug caused the event. Full disclaimer.

All Drugs Associated with Hepatotoxicity

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776 drugs have been associated with Hepatotoxicity in FAERS reports.

Drug Reports Deaths Hosp. Life-Threat.
METHOTREXATE 1,917 130 489 133
ACETAMINOPHEN 1,557 633 898 185
LEFLUNOMIDE 829 22 174 48
HYDROXYCHLOROQUINE 715 34 150 31
PREDNISONE 707 64 275 82
RITUXIMAB 702 77 211 46
ETANERCEPT 699 25 133 28
ADALIMUMAB 674 27 167 31
CYCLOPHOSPHAMIDE 632 98 155 72
SULFASALAZINE 613 26 166 33
RIBOCICLIB 585 49 113 65
TOCILIZUMAB 574 26 156 23
PEMBROLIZUMAB 542 55 140 21
DEXAMETHASONE 484 85 141 74
ABATACEPT 482 16 124 19
VINCRISTINE 474 69 132 67
DOXORUBICIN 468 58 132 62
CARBOPLATIN 452 58 108 21
LETROZOLE 416 29 80 51
CYTARABINE 366 73 91 49
PACLITAXEL 356 51 101 21
ISONIAZID 349 93 89 19
AZATHIOPRINE 329 42 97 35
NIVOLUMAB 324 46 130 22
INFLIXIMAB 316 26 72 21
DASATINIB 314 2 8 8
TOFACITINIB 313 23 119 22
ETOPOSIDE 302 55 66 46
VORICONAZOLE 298 51 106 32
PYRAZINAMIDE 279 59 94 18
TRASTUZUMAB 277 8 46 8
LINEZOLID 276 28 118 38
MYCOPHENOLATE MOFETIL 272 46 76 17
RIFAMPIN 271 78 88 16
PREDNISOLONE 263 45 87 35
OXALIPLATIN 258 15 50 23
BEDAQUILINE 254 8 44 13
CAPECITABINE 254 18 45 8
GOLIMUMAB 253 19 112 20
CERTOLIZUMAB PEGOL 249 18 126 20
IPILIMUMAB 234 28 113 17
ETHAMBUTOL 227 60 68 6
RISPERIDONE 224 0 197 1
MERCAPTOPURINE 213 24 68 24
IMATINIB 207 41 66 40
OLANZAPINE 207 11 185 6
QUETIAPINE 207 9 190 6
CISPLATIN 206 30 58 21
ATORVASTATIN 205 10 96 10
BEVACIZUMAB 203 28 30 3
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